Effects of administration route on pharmacokinetics of viloxazine in the rabbit

Methods Find Exp Clin Pharmacol. 1992 Mar;14(2):125-9.

Abstract

The absorption of viloxazine chlorhydrate was investigated in ten rabbits. Each animal received the drug (15 mg/kg) by three routes: intravenous, gastric and duodenal. Viloxazine plasma concentrations were low when administered by gastric and duodenal routes compared to those after intravenous injection. Concentrations to peak were 1-2 times higher after duodenal than gastric administration. Times to peak were 23.0 +/- 4.7 min after gastric administration and 9.5 +/- 5.4 min after duodenal administration. A better absorption of viloxazine after administration occurred in the duodenum than in the stomach; these results agree with viloxazine pKa = 8.13. The other pharmacokinetic parameters such as half-life, clearance and volume of distribution where the same irregardless of the administration route.

Publication types

  • Comparative Study

MeSH terms

  • Administration, Oral
  • Animals
  • Half-Life
  • Injections, Intravenous
  • Intestinal Absorption
  • Male
  • Rabbits
  • Tissue Distribution
  • Viloxazine / administration & dosage
  • Viloxazine / blood
  • Viloxazine / pharmacokinetics*

Substances

  • Viloxazine