Mouse Siglec-F and human Siglec-8 are functionally convergent paralogs that are selectively expressed on eosinophils and recognize 6'-sulfo-sialyl Lewis X as a preferred glycan ligand

Glycobiology. 2005 Nov;15(11):1125-35. doi: 10.1093/glycob/cwi097. Epub 2005 Jun 22.

Abstract

Mouse sialic acid-binding immunoglobulin-like lectin F (Siglec-F) is an eosinophil surface receptor, which contains an immunoreceptor tyrosine-based inhibitory motif (ITIM) in its cytoplasmic domain, implicating it as a regulator of cell signaling as documented for other siglecs. Here, we show that the sialoside sequence 6'-sulfo-sLe(X) (Neu5Acalpha2-3[6-SO4] Galbeta1-4[Fucalpha1-3]GlcNAc) is a preferred ligand for Siglec-F. In glycan array analysis of 172 glycans, recombinant Siglec-F-Fc chimeras bound with the highest avidity to 6'-sulfo-sLe X. Secondary analysis showed that related structures, sialyl-Lewis X (sLe X) and 6-sulfo-sLe X containing 6-GlcNAc-SO4 showed much lower binding avidity, indicating significant contribution of 6-Gal-SO4 on Siglec-F binding to 6'-sulfo-sLe x. The lectin activity of Siglec-F on mouse eosinophils was "masked" by endogenous cis ligands and could be unmasked by treatment with sialidase. Unmasked Siglec-F mediated mouse eosinophil binding and adhesion to multivalent 6'-sulfo-sLe X structure, and these interactions were inhibited by anti-Siglec-F monoclonal antibody (mAb). Although there is no clear-cut human ortholog of Siglec-F, Siglec-8 is encoded by a paralogous gene that is expressed selectively by human eosinophils and has recently been found to recognize 6'-sulfo-sLe X. These observations suggest that mouse Siglec-F and human Siglec-8 have undergone functional convergence during evolution and implicate a role for the interaction of these siglecs with their preferred 6'-sulfo-sLe X ligand in eosinophil biology.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Antibodies, Monoclonal / pharmacology
  • Antigens, CD / drug effects
  • Antigens, CD / genetics
  • Antigens, CD / physiology*
  • Antigens, Differentiation, B-Lymphocyte / drug effects
  • Antigens, Differentiation, B-Lymphocyte / genetics
  • Antigens, Differentiation, B-Lymphocyte / physiology*
  • Antigens, Differentiation, Myelomonocytic / drug effects
  • Antigens, Differentiation, Myelomonocytic / genetics
  • Antigens, Differentiation, Myelomonocytic / physiology*
  • CHO Cells
  • Cricetinae
  • Eosinophils / metabolism*
  • Humans
  • Lectins / drug effects
  • Lectins / genetics
  • Lectins / physiology*
  • Lewis X Antigen / analogs & derivatives
  • Ligands
  • Mice
  • Mice, Transgenic
  • Microscopy, Fluorescence
  • Neuraminidase / metabolism
  • Oligosaccharides / metabolism*
  • Polysaccharides / chemistry
  • Polysaccharides / metabolism*
  • Sialic Acid Binding Immunoglobulin-like Lectins
  • Sialyl Lewis X Antigen / analogs & derivatives

Substances

  • 6'-sulfated sialyl Lewis x
  • Antibodies, Monoclonal
  • Antigens, CD
  • Antigens, Differentiation, B-Lymphocyte
  • Antigens, Differentiation, Myelomonocytic
  • Lectins
  • Lewis X Antigen
  • Ligands
  • Oligosaccharides
  • Polysaccharides
  • SIGLEC8 protein, human
  • Sialic Acid Binding Immunoglobulin-like Lectins
  • Sialyl Lewis X Antigen
  • Siglecf protein, mouse
  • Neuraminidase