Regulation of myosin-IIA assembly and Mts1 binding by heavy chain phosphorylation

Biochemistry. 2005 May 10;44(18):6867-76. doi: 10.1021/bi0500776.

Abstract

Previous studies suggested that heavy chain phosphorylation regulates non-muscle myosin-II assembly in an isoform-specific manner, affecting the assembly of myosin-IIB, but not myosin-IIA. We re-examined the effects of heavy chain phosphorylation on myosin-IIA filament formation and also examined mts1 binding. We demonstrated that heavy chain phosphorylation by either protein kinase C (PKC) or casein kinase 2 (CK2) inhibits the assembly of myosin-IIA into filaments. PKC phosphorylation had no affect on mts1 binding, but CK2 phosphorylation decreased the affinity of mts1 for the myosin-IIA rod by approximately 6.5-fold. Mts1 destabilized PKC-phosphorylated myosin-IIA filaments and inhibited the assembly of myosin-IIA monomers with maximal inhibition of assembly and promotion of disassembly occurring at a molar ratio of one mts1 dimer per myosin-IIA rod. At this molar ratio, mts1 only weakly disassembled CK2-phosphorylated myosin-IIA filaments and weakly inhibited the assembly of CK2-phosphorylated myosin-IIA monomers. These observations demonstrate that CK2 phosphorylation of the myosin-IIA heavy chain protects against mts1-induced filament disassembly and inhibition of assembly, and suggest that heavy chain phosphorylation provides an additional level of regulation for the mts1-myosin-IIA interaction.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Actin Cytoskeleton / enzymology
  • Actin Cytoskeleton / metabolism
  • Casein Kinase II / chemistry
  • Casein Kinase II / metabolism
  • Computer Simulation
  • Humans
  • Models, Molecular
  • Myosin Heavy Chains / antagonists & inhibitors
  • Myosin Heavy Chains / chemistry
  • Myosin Heavy Chains / metabolism*
  • Nonmuscle Myosin Type IIA / antagonists & inhibitors
  • Nonmuscle Myosin Type IIA / chemistry
  • Nonmuscle Myosin Type IIA / metabolism*
  • Peptide Fragments / antagonists & inhibitors
  • Peptide Fragments / chemistry
  • Peptide Fragments / metabolism
  • Phosphorylation
  • Polymers / chemistry
  • Polymers / metabolism
  • Protein Binding
  • Protein Isoforms / antagonists & inhibitors
  • Protein Isoforms / chemistry
  • Protein Isoforms / metabolism
  • Protein Kinase C / chemistry
  • Protein Kinase C / metabolism
  • Protein Processing, Post-Translational / physiology*
  • Protein Structure, Tertiary
  • S100 Calcium-Binding Protein A4
  • S100 Proteins / chemistry
  • S100 Proteins / metabolism*

Substances

  • Peptide Fragments
  • Polymers
  • Protein Isoforms
  • S100 Calcium-Binding Protein A4
  • S100 Proteins
  • S100A4 protein, human
  • Casein Kinase II
  • Protein Kinase C
  • Nonmuscle Myosin Type IIA
  • Myosin Heavy Chains