Transcriptional regulation of a metastasis suppressor gene by Tip60 and beta-catenin complexes

Nature. 2005 Apr 14;434(7035):921-6. doi: 10.1038/nature03452.

Abstract

Defining the molecular strategies that integrate diverse signalling pathways in the expression of specific gene programmes that are critical in homeostasis and disease remains a central issue in biology. This is particularly pertinent in cancer biology because downregulation of tumour metastasis suppressor genes is a common occurrence, and the underlying molecular mechanisms are not well established. Here we report that the downregulation of a metastasis suppressor gene, KAI1, in prostate cancer cells involves the inhibitory actions of beta-catenin, along with a reptin chromatin remodelling complex. This inhibitory function of beta-catenin-reptin requires both increased beta-catenin expression and recruitment of histone deacetylase activity. The coordinated actions of beta-catenin-reptin components that mediate the repressive state serve to antagonize a Tip60 coactivator complex that is required for activation; the balance of these opposing complexes controls the expression of KAI1 and metastatic potential. The molecular mechanisms underlying the antagonistic regulation of beta-catenin-reptin and the Tip60 coactivator complexes for the metastasis suppressor gene, KAI1, are likely to be prototypic of a selective downregulation strategy for many genes, including a subset of NF-kappaB target genes.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Acetyltransferases / genetics
  • Acetyltransferases / metabolism*
  • Animals
  • Antigens, CD / genetics*
  • Cell Line, Tumor
  • Chromatin Assembly and Disassembly
  • Collagen
  • Cytoskeletal Proteins / metabolism*
  • Down-Regulation / genetics
  • Drug Combinations
  • Gene Expression Regulation, Neoplastic / genetics*
  • Histone Acetyltransferases
  • Humans
  • Kangai-1 Protein
  • Laminin
  • Lysine Acetyltransferase 5
  • Male
  • Membrane Glycoproteins / genetics*
  • Mice
  • NF-kappa B / metabolism
  • Neoplasm Metastasis / genetics*
  • Neoplasm Transplantation
  • Promoter Regions, Genetic / genetics
  • Prostatic Neoplasms / genetics*
  • Prostatic Neoplasms / metabolism
  • Proteoglycans
  • Proto-Oncogene Proteins / genetics*
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • Trans-Activators / metabolism*
  • Transcription, Genetic / genetics*
  • beta Catenin

Substances

  • Antigens, CD
  • CD82 protein, human
  • CTNNB1 protein, human
  • CTNNB1 protein, mouse
  • Cd82 antigen, mouse
  • Cytoskeletal Proteins
  • Drug Combinations
  • Kangai-1 Protein
  • Laminin
  • Membrane Glycoproteins
  • NF-kappa B
  • Proteoglycans
  • Proto-Oncogene Proteins
  • RNA, Messenger
  • Trans-Activators
  • beta Catenin
  • matrigel
  • Collagen
  • Acetyltransferases
  • Histone Acetyltransferases
  • KAT5 protein, human
  • Lysine Acetyltransferase 5