D-beta-hydroxybutyrate is neuroprotective against hypoxia in serum-free hippocampal primary cultures

J Neurosci Res. 2005 May 15;80(4):501-9. doi: 10.1002/jnr.20464.

Abstract

Hypoxia decreased survival of cultured rat primary hippocampal neurons in a time dependent manner. Addition of 4 mM Na D-beta-hydroxybutyrate (bHB), a ketone body, protected the cells for 2 hr and maintained the increase in survival compared to that of controls for up to 6 hr. Trypan blue exclusion indicated that acute cell death was reduced markedly after 2-hr exposure to hypoxia in the bHB-treated group. The presence of bHB also decreased the number of neurons exhibiting condensed nuclei visualized by propidium iodide, indicative of apoptosis. The mitochondrial transmembrane potential (Em/c) was maintained for up to 2 hr exposure to hypoxia in the bHB-treated group, whereas the potential in the control group was decreased. Furthermore, cytochrome C release, caspase-3 activation, and poly (ADP-ribose) polymerase (PARP) cleavage were decreased in the bHB-treated group for the first 2 hr of exposure. These findings indicate that ketone bodies may be a candidate for widening the therapeutic window before thrombolytic therapy and at the same time decreasing apoptotic damage in the ischemic penumbra.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3-Hydroxybutyric Acid / pharmacology*
  • Animals
  • Caspase 3
  • Caspases / metabolism
  • Cell Hypoxia / drug effects
  • Cell Survival / drug effects
  • Cells, Cultured
  • Culture Media, Serum-Free / pharmacology
  • Cytochromes c / metabolism
  • Embryo, Mammalian
  • Glial Fibrillary Acidic Protein / metabolism
  • Hippocampus / cytology*
  • Immunohistochemistry / methods
  • Membrane Potentials / drug effects
  • Microtubule-Associated Proteins / metabolism
  • Mitochondria / drug effects
  • Neurons / drug effects*
  • Neurons / metabolism
  • Neuroprotective Agents / pharmacology*
  • Poly(ADP-ribose) Polymerases / metabolism
  • Propidium
  • Rats
  • Rats, Wistar
  • Statistics, Nonparametric
  • Time Factors
  • Trypan Blue

Substances

  • Culture Media, Serum-Free
  • Glial Fibrillary Acidic Protein
  • MAP2 protein, rat
  • Microtubule-Associated Proteins
  • Neuroprotective Agents
  • Propidium
  • Cytochromes c
  • Poly(ADP-ribose) Polymerases
  • Casp3 protein, rat
  • Caspase 3
  • Caspases
  • Trypan Blue
  • 3-Hydroxybutyric Acid