pH-dependent intraluminal organization of mucin granules in live human mucous/goblet cells

J Biol Chem. 2005 Apr 29;280(17):16868-81. doi: 10.1074/jbc.M413289200. Epub 2005 Feb 17.

Abstract

To study the mechanism of gel-forming mucin packaging within mucin granules, we generated human mucous/goblet cells stably expressing a recombinant MUC5AC domain fused to green fluorescent protein (GFP). The fusion protein, named SHGFP-MUC5AC/CK, accumulated in the granules together with native MUC5AC. Inhibition of protein synthesis or disorganization of the Golgi complex did not result in diminished intragranular SHGFP-MUC5AC/CK signals, consistent with long-term storage of the fusion protein. However, SHGFP-MUC5AC/CK was rapidly discharged from the granules upon incubation of the cells with ATP, an established mucin secretagogue. Several criteria indicated that SHGFP-MUC5AC/CK was not covalently linked to endogenous MUC5AC. Analysis of fluorescence recovery after photobleaching suggested that the intragranular SHGFP-MUC5AC/CK mobile fraction and mobility were significantly lower than in the endoplasmic reticulum lumen. Incubation of the cells with bafilomycin A1, a specific inhibitor of the vacuolar H+-ATPase, did not alter the fusion protein mobility, although it significantly increased (approximately 20%) the intragranular SHGFP-MUC5AC/CK mobile fraction. In addition, the granules in bafilomycin-incubated cells typically exhibited a heterogeneous intraluminal distribution of the fluorescent fusion protein. These results are consistent with a model of mucin granule intraluminal organization with two phases: a mobile phase in which secretory proteins diffuse as in the endoplasmic reticulum lumen but at a lower rate and an immobile phase or matrix in which proteins are immobilized by noncovalent pH-dependent interactions. An intraluminal acidic pH, maintained by the vacuolar H+-ATPase, is one of the critical factors for secretory protein binding to the immobile phase and also for its organization.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenosine Triphosphatases / chemistry
  • Adenosine Triphosphate / chemistry
  • Amino Acid Sequence
  • Animals
  • COS Cells
  • Calcium / metabolism
  • Cloning, Molecular
  • DNA, Complementary / metabolism
  • Endoplasmic Reticulum / metabolism
  • Fluorescence Recovery After Photobleaching
  • Goblet Cells / metabolism*
  • Green Fluorescent Proteins / metabolism
  • Humans
  • Hydrogen-Ion Concentration
  • Macrolides / pharmacology
  • Microscopy, Electron
  • Molecular Sequence Data
  • Mucin 5AC
  • Mucins / chemistry*
  • Mucins / metabolism
  • Phenotype
  • Protein Binding
  • Protein Structure, Tertiary
  • Recombinant Fusion Proteins / metabolism
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / metabolism
  • Signal Transduction
  • Time Factors

Substances

  • DNA, Complementary
  • MUC5AC protein, human
  • Macrolides
  • Mucin 5AC
  • Mucins
  • Recombinant Fusion Proteins
  • Recombinant Proteins
  • bafilomycin A
  • Green Fluorescent Proteins
  • bafilomycin A1
  • Adenosine Triphosphate
  • Adenosine Triphosphatases
  • Calcium