Leptin and post-prandial satiety: acute central leptin more potently reduces meal frequency than meal size in the rat

Psychopharmacology (Berl). 2005 Jan;177(3):324-35. doi: 10.1007/s00213-004-1952-1. Epub 2004 Jul 27.

Abstract

Rationale: Many attempts to understand ingestion have sought to clarify the control of meals. Little is known about the effects of the anorexogenic hormone leptin on meal patterning.

Objective: The present study sought to perform a dose-response analysis of the effects of acute central leptin administration on meal patterning using a validated, objective meal definition and to compare these results to those obtained with a previously used, subjective meal definition.

Methods: To validate the objective meal definition pharmacologically, the microstructural effects of the well-studied compound fenfluramine (SC 0, 1, 2, 4 mg/kg) on spontaneous nocturnal intake were determined in mature, non-deprived male Wistar rats (n=8) using a full Latin square design. The effects of intracerebroventricular leptin administration (0, 0.3, 1, 3, 6.25 microg; n=10) were also examined, and perceived meal patterns obtained from the objective and subjective definitions were compared.

Results: Fenfluramine reduced meal size and eating rate at doses that did not reduce meal frequency or duration. In contrast, comparably anorectic doses of leptin had potent post-meal satiety-like effects, reducing meal frequency and prolonging the intermeal interval without reducing average meal size, a finding opposite to that suggested by the previously used subjective meal definition. Unlike comparably and more anorectic doses of fenfluramine, leptin non-specifically reduced both prandial and non-prandial drinking.

Conclusions: Acute increases in central leptin levels may potently augment post-prandial satiety and influence body-fluid homeostasis. The results reveal unappreciated central modes of action for the ob protein which qualitatively differ from the intra-meal satiating-like effects of fenfluramine.

Publication types

  • Comparative Study
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Appetite Regulation / drug effects*
  • Appetite Regulation / physiology
  • Circadian Rhythm / drug effects
  • Circadian Rhythm / physiology
  • Dose-Response Relationship, Drug
  • Drinking / drug effects
  • Drinking / physiology
  • Eating / drug effects
  • Eating / physiology
  • Fenfluramine / administration & dosage
  • Fenfluramine / pharmacokinetics
  • Injections, Intraventricular
  • Injections, Subcutaneous
  • Leptin / administration & dosage
  • Leptin / metabolism
  • Leptin / pharmacokinetics*
  • Male
  • Postprandial Period / drug effects*
  • Postprandial Period / physiology
  • Psychopharmacology / methods
  • Rats
  • Rats, Wistar
  • Satiety Response / drug effects*
  • Satiety Response / physiology

Substances

  • Leptin
  • Fenfluramine