Erythropoietin production rate in phlebotomy-induced acute anemia

Biopharm Drug Dispos. 2004 Dec;25(9):389-97. doi: 10.1002/bdd.424.

Abstract

Objective: To estimate the rate of erythropoietin (EPO) production under physiological, conditions and to examine the regulatory mechanism of EPO production in response to acute phlebotomy-induced anemia.

Methods: Six sheep each underwent two phlebotomies in which the hemoglobin (Hb) was reduced to 3-4 g/dl over 4-5 h. The EPO plasma level, reticulocytes, Hb and EPO clearance were followed by frequent blood sampling. The EPO production rate was determined by a semi-parametric method based on a disposition decomposition analysis that accounts for the nonlinear disposition kinetics of EPO and corrects for time-dependent changes in the clearance.

Results: The controlled drop in hemoglobin resulted in an abrupt increase in the plasma EPO concentration (peak level 812+/-40 mU/ml, mean+/-CV%) that was followed by a rapid drop 2-4 days after the phlebotomy at a time when the sheep were still anemic (Hb=4.3+/-16 g/dl). The EPO production rate at baseline was 43+/-52 U/day/kg and the amounts of EPO produced over an 8 day period resulting from the first and second phlebotomy were 2927+/-40 U/kg and 3012+/-31 U/kg, respectively.

Conclusions: The rapid reduction in the EPO plasma level observed 2-4 days following the phlebotomy cannot be explained solely by the increase in EPO clearance but also by a reduction in EPO production.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Acute Disease
  • Anemia / blood*
  • Anemia / etiology
  • Animals
  • Erythropoietin / biosynthesis*
  • Erythropoietin / blood*
  • Hemoglobins / metabolism
  • Linear Models
  • Models, Biological
  • Nonlinear Dynamics
  • Phlebotomy / adverse effects*
  • Sheep
  • Time Factors

Substances

  • Hemoglobins
  • Erythropoietin