Safety and adverse effects associated with raloxifene: multiple outcomes of raloxifene evaluation

Obstet Gynecol. 2004 Oct;104(4):837-44. doi: 10.1097/01.AOG.0000137349.79204.b8.

Abstract

Objective: To examine the effect of raloxifene on major adverse events that occur with postmenopausal estrogen therapy or tamoxifen.

Methods: The Multiple Outcomes of Raloxifene Evaluation, a multicenter, randomized, double-blind trial, enrolled 7,705 postmenopausal women with osteoporosis. Women were randomly assigned to raloxifene 60 mg/d or 120 mg/d or placebo. Outcomes included venous thromboembolism, cataracts, gallbladder disease, and endometrial hyperplasia or cancer.

Results: During a mean follow-up of 3.3 years, raloxifene was associated with an increased risk for venous thromboembolism (relative risk [RR] 2.1; 95% confidence interval [CI] 1.2-3.8). The excess event rate was 1.8 per 1,000 woman-years (95% CI -0.5-4.1), and the number needed to treat to cause 1 event was 170 (95% CI 100-582) over 3.3 years. Risk in the raloxifene group was higher than in the placebo group for the first 2 years, but decreased to about the same rate as in the placebo group thereafter. Raloxifene did not increase risk for cataracts (RR 0.9; 95% CI 0.8-1.1), gallbladder disease (RR 1.0; 95% CI 0.7-1.3), endometrial hyperplasia (RR 1.3; 95% CI 0.4-5.1), or endometrial cancer (RR 0.9; 95% CI 0.3-2.7).

Conclusion: Raloxifene was associated with an increased risk for venous thromboembolism, but there was no increased risk for cataracts, gallbladder disease, endometrial hyperplasia, or endometrial cancer.

Level of evidence: I

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Double-Blind Method
  • Female
  • Humans
  • Incidence
  • Middle Aged
  • Multicenter Studies as Topic
  • Osteoporosis, Postmenopausal / drug therapy*
  • Raloxifene Hydrochloride / adverse effects*
  • Raloxifene Hydrochloride / therapeutic use
  • Selective Estrogen Receptor Modulators / adverse effects*
  • Selective Estrogen Receptor Modulators / therapeutic use
  • United States / epidemiology
  • Venous Thrombosis / chemically induced*
  • Venous Thrombosis / epidemiology*

Substances

  • Selective Estrogen Receptor Modulators
  • Raloxifene Hydrochloride