A facile synthesis of C2,N3-disubstituted-4-quinazolone

J Org Chem. 2004 Sep 17;69(19):6474-7. doi: 10.1021/jo049118e.

Abstract

A simple and efficient methodology for the synthesis of C(2),N(3)-disubstituted-4 quinazolones from anilines and N-acylanthranilic acids was developed. The new cyclization conditions are much milder than any other reported protocols and resulted in excellent yields (87-98%) without chromatography.