Influence of some convulsant agents on the protective activity of a novel antiepileptic drug, felbamate, against maximal electroshock in mice

Pol J Pharmacol. 2003 Jul-Aug;55(4):649-53.

Abstract

The aim of this study was to evaluate effects of strychnine, as well as bicuculline and picrotoxin on the anticonvulsant action of felbamate against maximal electroshock (MES)-induced seizures in mice. Strychnine (up to 0.5 mg/kg), bicuculline (up to 2 mg/kg) and picrotoxin (3 mg/kg) did not affect the seizure threshold. However, strychnine (0.25-0.5 mg/kg) and picrotoxin (3 mg/kg) impaired the protective activity of felbamate against MES. It may be concluded that GABAergic inhibition and strychnine-insensitive glycine receptor-mediated events may contribute to the anticonvulsant activity of felbamate.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Anticonvulsants / pharmacology*
  • Bicuculline / pharmacology
  • Convulsants / pharmacology*
  • Dose-Response Relationship, Drug
  • Drug Interactions
  • Electroshock
  • Felbamate
  • Male
  • Mice
  • Neuroprotective Agents / pharmacology
  • Phenylcarbamates
  • Picrotoxin / pharmacology
  • Propylene Glycols / pharmacology*
  • Rats
  • Seizures / etiology
  • Seizures / prevention & control*
  • Strychnine / pharmacology

Substances

  • Anticonvulsants
  • Convulsants
  • Neuroprotective Agents
  • Phenylcarbamates
  • Propylene Glycols
  • Picrotoxin
  • Strychnine
  • Felbamate
  • Bicuculline