Prenoids and palmitate: lipids that control the biological activity of Ras proteins

Semin Cancer Biol. 1992 Aug;3(4):179-88.

Abstract

Ras proteins can be modified by two types of lipids--an isoprenoid and the fatty acid palmitate. These lipids help the otherwise cytoplasmic Ras protein to interact with the plasma membrane of a cell. The biological consequences of this association between Ras and membranes are dramatic, and can alter a cell's behavior from normal growth into malignancy. The scope and limits of our knowledge of the steps, structures and enzymes involved in this molecular transformation from soluble inactivity to membrane-bound potency are offered below. The prospects of regulating Ras function by controlling its intracellular location provides a tantalizing opportunity to translate research into a novel therapeutic reality.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.
  • Review

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Gene Expression Regulation / physiology*
  • Genes, ras / physiology*
  • Molecular Sequence Data
  • Palmitic Acid
  • Palmitic Acids / metabolism*
  • Polyisoprenyl Phosphates / metabolism*
  • Protein Prenylation / physiology
  • Saccharomyces cerevisiae

Substances

  • Palmitic Acids
  • Polyisoprenyl Phosphates
  • Palmitic Acid