R5020 enhances PGE2 stimulated steroidogenesis in cultured rat granulosa cells

Rev Esp Fisiol. 1992 Sep;48(3):167-70.

Abstract

Progesterone biosynthesis and metabolization to 20 alpha-hydroxyprogesterone was stimulated in granulosa cells cultured in the presence of 20 ng/ml of follicle stimulating hormone (FSH) or increasing concentrations of PGE2 (10(-9)-10(-7)M). Concurrent treatment with the synthetic progestin R5020 (10(-6) M) enhanced the FSH or PGE2 stimulated progesterone and 20 alpha-hydroxyprogesterone accumulation in culture media, as well as delta 5-3 beta-hydroxysteroid dehydrogenase activity in granulosa cell homogenates. These findings may represent another example of an autocrine control mechanism in which the steroidogenic product of the granulosa cell exerts an ultra-short loop regulation of its own production.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 20-alpha-Dihydroprogesterone / biosynthesis
  • 3-Hydroxysteroid Dehydrogenases / metabolism
  • Animals
  • Cells, Cultured
  • Dinoprostone / pharmacology*
  • Drug Synergism
  • Female
  • Follicle Stimulating Hormone / pharmacology
  • Granulosa Cells / drug effects*
  • Granulosa Cells / metabolism
  • Progesterone / biosynthesis*
  • Promegestone / pharmacology*
  • Rats
  • Rats, Sprague-Dawley
  • Stimulation, Chemical

Substances

  • 20-alpha-Dihydroprogesterone
  • Progesterone
  • Follicle Stimulating Hormone
  • Promegestone
  • 3-Hydroxysteroid Dehydrogenases
  • delta(5)-3 beta-hydroxysteroid dehydrogenase
  • Dinoprostone