Effects of a new antiarrhythmic drug, SD-3212, on canine ventricular arrhythmia models

Jpn Heart J. 1992 Nov;33(6):851-61. doi: 10.1536/ihj.33.851.

Abstract

The antiarrhythmic effects of a new antiarrhythmic agent, SD-3212, (-)-(S)-3,4-Dihydro-2-[5-methoxy-2-[3-[N-methyl-N-[2-[(3,4- methylene dioxy)phenoxy]ethyl]amino]propoxy]phenyl]-4-methyl-3-oxo-2H-1, 4-benzothiazine hydrogen fumarate, were investigated using canine models of ventricular arrhythmias, i.e. spontaneously occurring digitalis-, two-stage coronary ligation- and adrenaline-induced arrhythmias. SD-3212 suppressed adrenaline-induced arrhythmia and showed some antiarrhythmic effect on digitalis- and 48 hr coronary ligation-arrhythmias. These results indicate that SD-3212 has antiarrhythmic effects common among class IV antiarrhythmic drugs and also has additional efficacy common among class I antiarrhythmic drugs, thus when considering the level of experimental arrhythmias it somewhat resembles propafenone. It may therefore become a clinically useful antiarrhythmic drug among typical class I or class IV antiarrhythmic drugs.

MeSH terms

  • Animals
  • Anti-Arrhythmia Agents / pharmacology*
  • Arrhythmias, Cardiac / chemically induced
  • Arrhythmias, Cardiac / etiology
  • Arrhythmias, Cardiac / physiopathology*
  • Coronary Vessels
  • Digitalis
  • Dogs
  • Epinephrine
  • Female
  • Ligation
  • Male
  • Osmolar Concentration
  • Plants, Medicinal
  • Plants, Toxic
  • Thiazoles / blood
  • Thiazoles / pharmacology*

Substances

  • Anti-Arrhythmia Agents
  • Thiazoles
  • sesamodil
  • Epinephrine