Synthesis of amide compounds of ferulic acid, and their stimulatory effects on insulin secretion in vitro

Bioorg Med Chem. 2003 Aug 15;11(17):3807-13. doi: 10.1016/s0968-0896(03)00280-3.

Abstract

We prepared amide compounds which were derived from ferulic acid using various amines, and investigated their stimulatory effects on insulin secretion using rat pancreatic RIN-5F cells. Most of these compounds exhibited significant promotion of the insulin-release at a concentration of 10 microM and in particular, the amides having n-butyl, n-pentyl, pyrrolidine, and piperidine groups showed high activity.

MeSH terms

  • Amides / chemical synthesis*
  • Amides / pharmacology*
  • Animals
  • Cell Survival
  • Coumaric Acids / chemical synthesis
  • Coumaric Acids / chemistry*
  • Coumaric Acids / pharmacology
  • Dose-Response Relationship, Drug
  • Insulin / biosynthesis*
  • Rats

Substances

  • Amides
  • Coumaric Acids
  • Insulin
  • ferulic acid