ATP-binding is stabilized by a stacking interaction within the binding site of Na+/K+ -ATPase

Biochem Biophys Res Commun. 2003 Jun 27;306(2):416-20. doi: 10.1016/s0006-291x(03)00946-x.

Abstract

Site-directed mutagenesis was applied to modify phenylalanines (Phe(475)Trp, Phe(548)Tyr, and both) to generate mutants on the basis of molecular modeling of the ATP-binding domain of Na(+)/K(+)-ATPase, in order to characterize the forces that stabilize ATP in its binding pocket. Each of the mutants was examined by Raman difference spectroscopy, i.e., as a difference between the spectrum of the domain with and without bound ATP. It was shown that Phe(475) plays a key role in stabilizing ATP-binding by a stacking interaction. Phe(548) co-stabilizes ATP on the opposite site of the binding pocket and its type of interaction with ATP-binding differs from that of Phe(475).

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Triphosphate / metabolism*
  • Animals
  • Binding Sites
  • Chromatography, High Pressure Liquid
  • Mice
  • Models, Molecular
  • Mutagenesis, Site-Directed
  • Mutation
  • Phenylalanine / chemistry
  • Protein Binding
  • Protein Structure, Secondary
  • Protein Structure, Tertiary
  • Sodium-Potassium-Exchanging ATPase / chemistry*
  • Sodium-Potassium-Exchanging ATPase / metabolism
  • Spectrum Analysis, Raman

Substances

  • Phenylalanine
  • Adenosine Triphosphate
  • Sodium-Potassium-Exchanging ATPase