A thrombin-cross-reactive anticardiolipin antibody binds to and inhibits the anticoagulant function of activated protein C

Arthritis Rheum. 2003 Jun;48(6):1622-30. doi: 10.1002/art.10983.

Abstract

Objective: To test the hypotheses that some thrombin-reactive anticardiolipin antibodies (aCL) may bind to protein C (PC) and/or activated PC (APC), and that some of the PC- and APC-reactive aCL may inhibit PC activation and/or the function of APC.

Methods: We studied the reactivity of patient-derived monoclonal aCL with PC and APC. We examined the effects of the reactive antibodies on PC activation and on the activity of APC in plasma coagulation.

Results: Five of 5 patient-derived, thrombin-reactive monoclonal aCL bound to PC and APC. In addition, 1 patient-derived monoclonal antiprothrombin antibody (APT) that displayed aCL activity and reacted with thrombin also bound to PC and APC. Of these 6 PC- and APC-reactive aCL/APT, all failed to inhibit PC activation, but 1 (CL15) shortened the plasma coagulation time in the presence of exogenous APC and thus inhibited the anticoagulant function of APC.

Conclusion: Most of the thrombin-reactive aCL in patients with antiphospholipid syndrome may bind to PC and APC. Of the APC-reactive aCL, some (like CL15) may inhibit the anticoagulant function of APC and are thus likely to be prothrombotic in the host.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Antibodies, Anticardiolipin / immunology*
  • Antibodies, Monoclonal / immunology
  • Antibody Affinity
  • Anticoagulants / immunology*
  • Binding Sites, Antibody
  • Cross Reactions / immunology
  • Dose-Response Relationship, Immunologic
  • Humans
  • Models, Molecular
  • Molecular Sequence Data
  • Protein C / chemistry
  • Protein C / immunology*
  • Protein C Inhibitor / immunology*
  • Thrombin / chemistry
  • Thrombin / immunology*

Substances

  • Antibodies, Anticardiolipin
  • Antibodies, Monoclonal
  • Anticoagulants
  • Protein C
  • Protein C Inhibitor
  • Thrombin