The protective mechanism of magnolol, a Chinese herb drug, against warm ischemia-reperfusion injury of rat liver

J Surg Res. 2003 Apr;110(2):378-82. doi: 10.1016/s0022-4804(03)00034-9.

Abstract

Background: Cell apoptosis following warm ischemia-reperfusion injury is a major concern in clinical issues such as organ transplantation, trauma, and cardiogenic shock. The purpose of this study was to evaluate the possible role of magnolol, a Chinese herb drug, in apoptotic injury and the kinetic expression of apoptotic-related genes in rat livers subjected to warm ischemia-reperfusion (WI/R).

Materials and methods: Three weeks prior to the experiment 10 rats underwent a portosystemic shunt operation according to Bengmerk's method. The rats were divided into three groups. Group 1 (GI) was the control group, Group 2 (GII) and Group 3 (GIII) the magnolol-treated groups. GI and GII were subjected to 2 h and GIII to 3 h of WI/R by clamping the portal vein and hepatic artery under ether anesthesia.

Results: Results show that all the control rats died after 2 h WI/R. Apoptotic cells were detected under microscopy as well as by DNA assay. Magnolol-treated groups tolerated warm ischemia-reperfusion for 2 h and significantly less apoptotic cells were observed (198 +/- 22 vs 42.6 +/- 28). But magnolol-treated rats could not tolerate 3 h warm ischemia-reperfusion. RT-PCR of liver tissue shows that there is an upregulated expression of the anti-apoptotic Bcl-xL gene and suppression of the Bcl-xS gene in GII.

Conclusion: Magnolol has an anti-apoptotic effect and protects the liver against WI/R for 2 h but not for 3 h through upregulation of the anti-apoptotic Bcl-XL gene and suppression of the Bcl-xS gene.

Publication types

  • Evaluation Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis / drug effects*
  • Apoptosis / genetics
  • Biphenyl Compounds / pharmacology*
  • Drugs, Chinese Herbal / pharmacology
  • Enzyme Inhibitors / pharmacology*
  • Gene Expression Regulation
  • Lignans*
  • Liver / blood supply*
  • Liver / drug effects*
  • Liver / physiopathology
  • Models, Animal
  • Nitric Oxide Synthase / antagonists & inhibitors*
  • Proto-Oncogene Proteins c-bcl-2 / genetics
  • Proto-Oncogene Proteins c-bcl-2 / physiology
  • Rats
  • Reperfusion Injury / drug therapy*
  • Reperfusion Injury / genetics
  • Reperfusion Injury / physiopathology
  • bcl-X Protein

Substances

  • Bcl2l1 protein, rat
  • Biphenyl Compounds
  • Drugs, Chinese Herbal
  • Enzyme Inhibitors
  • Lignans
  • Proto-Oncogene Proteins c-bcl-2
  • bcl-X Protein
  • magnolol
  • Nitric Oxide Synthase