D-alanine piperazine-amides: novel non-imidazole antagonists of the histamine H3 receptor

Inflamm Res. 2003 Apr:52 Suppl 1:S47-8. doi: 10.1007/s000110300049.
No abstract available

MeSH terms

  • Alanine / chemistry
  • Amides / chemistry
  • Animals
  • Binding, Competitive / drug effects
  • Histamine Antagonists / chemical synthesis*
  • Histamine Antagonists / pharmacology*
  • Humans
  • Indicators and Reagents
  • Kinetics
  • Piperazines / chemical synthesis*
  • Piperazines / pharmacology*
  • Rats
  • Receptors, Histamine H3 / drug effects*
  • Recombinant Proteins / metabolism

Substances

  • 4-((3-(4-(2-aminopropanoyl)-1-piperazinyl)propoxy)phenyl)cyclopropylmethanone
  • Amides
  • Histamine Antagonists
  • Indicators and Reagents
  • Piperazines
  • Receptors, Histamine H3
  • Recombinant Proteins
  • Alanine