Powdered cellulose as excipient for extrusion-spheronization pellets of a cohesive hydrophobic drug

Eur J Pharm Biopharm. 2003 May;55(3):291-5. doi: 10.1016/s0939-6411(03)00032-8.

Abstract

This study compared a powdered cellulose (PC) and a microcrystalline cellulose (MCC) as sole excipients in the preparation of furosemide pellets by extrusion-spheronization. Pellets prepared with PC and 25 or 50% furosemide showed smaller mean size, a broader particle size distribution, similar sphericity, greater surface roughness and higher friability than equivalent pellets prepared with MCC. Furosemide release rate was markedly higher from PC pellets, which may be attributable to their higher micropore volume.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cellulose / chemistry
  • Cellulose / pharmacokinetics*
  • Chemistry, Pharmaceutical
  • Drug Implants
  • Excipients / chemistry
  • Excipients / pharmacokinetics*
  • Hydrophobic and Hydrophilic Interactions*
  • Powders

Substances

  • Drug Implants
  • Excipients
  • Powders
  • Cellulose