Identification of a PU.1-IRF4 protein interaction surface predicted by chemical exchange line broadening

Proc Natl Acad Sci U S A. 2003 Jan 21;100(2):511-6. doi: 10.1073/pnas.0136910100. Epub 2003 Jan 7.

Abstract

Relaxation values reflecting residue-specific line broadening revealed amino acids in the DNA-binding domain of PU.1 on a surface potentially involved in protein-protein interactions. Mutation of these amino acids did not cause protein unfolding but destabilized PU.1-DNA binding. Addition of IFN response factor 4 to form the ternary complex recovered binding stability. Fluorescence quenching experiments proved that this surface of PU.1 interacts with IFN response factor 4 during binding. Our results provide evidence that residues that display increased conformational exchange can be used to predict areas of protein-protein interactions.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Binding Sites
  • DNA / metabolism
  • DNA-Binding Proteins / chemistry*
  • Fluorescence
  • Interferon Regulatory Factors
  • Mutation
  • Protein Conformation
  • Proto-Oncogene Proteins / chemistry*
  • Trans-Activators / chemistry*
  • Transcription Factors / chemistry*

Substances

  • DNA-Binding Proteins
  • Interferon Regulatory Factors
  • Proto-Oncogene Proteins
  • Trans-Activators
  • Transcription Factors
  • interferon regulatory factor-4
  • proto-oncogene protein Spi-1
  • DNA