Unusual cyanide bindings to a heme-regulated phosphodiesterase from Escherichia coli: effect of Met95 mutations

Biochem Biophys Res Commun. 2002 Nov 29;299(2):169-72. doi: 10.1016/s0006-291x(02)02621-9.

Abstract

In order to understand heme environment of a heme-regulated phosphodiesterase (Ec DOS), the binding behavior of cyanide to the Fe (III) complex was examined. Interestingly, the rate of cyanide binding to full-length Ec DOS was unusually slow with k(on)=0.0022mM(-1)s(-1), while the rate for the isolated heme domain of Ec DOS (0.045mM(-1)s(-1)) was 20-fold higher. Ala and Leu mutations at Met95, which has been suggested to be a heme axial ligand, increased the k(on) rate 11- and 8-fold, respectively, and dramatically decreased the cyanide dissociation rate from the isolated heme domain. His mutation at Met95, on the other hand, caused a 17-fold decrease in the k(on) value. We discuss the unusual cyanide binding behavior and the role of Met95 in controlling cyanide binding.

MeSH terms

  • Azides / metabolism
  • Cyanides / metabolism*
  • Escherichia coli / enzymology*
  • Fluorides / metabolism
  • Heme / metabolism*
  • Imidazoles / metabolism
  • Iron / metabolism
  • Kinetics
  • Methionine / genetics*
  • Mutagenesis, Site-Directed
  • Mutation
  • Phosphoric Diester Hydrolases / chemistry
  • Phosphoric Diester Hydrolases / genetics
  • Phosphoric Diester Hydrolases / metabolism*
  • Protein Binding
  • Protein Structure, Tertiary
  • Spectrophotometry

Substances

  • Azides
  • Cyanides
  • Imidazoles
  • Heme
  • Methionine
  • Iron
  • Phosphoric Diester Hydrolases
  • Fluorides