Organisation of G-protein-coupled receptor signalling complexes by scaffolding proteins

Curr Opin Pharmacol. 2002 Oct;2(5):581-6. doi: 10.1016/s1471-4892(02)00203-5.

Abstract

Signalling by receptors coupled to heterotrimeric G proteins primarily involves intermediates (G-protein subunits and second messengers) that can reach their targets by diffusion either through the cytosol or within the plane of the membrane. However, in many cases additional proteins have been identified which, by providing a scaffold, link several components of a signal transduction pathway in order to control speed and specificity of signalling. Scaffolding proteins such as PSD-95 or shank/ProSAP proteins organise rather large signalling complexes. Recent proteomic approaches have now been used to study the molecular composition of receptor complexes in detail, for example glutamate receptors and 5HT(2C) receptors, providing a much more complicated picture of G-protein-coupled receptor signalling than previously anticipated.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Carrier Proteins / chemistry
  • GTP-Binding Proteins / chemistry
  • GTP-Binding Proteins / metabolism*
  • Homer Scaffolding Proteins
  • Humans
  • Insecta
  • Neuropeptides / chemistry
  • Proteomics
  • Receptor Cross-Talk / physiology
  • Receptors, Drug / chemistry
  • Receptors, Drug / metabolism*
  • Receptors, Glutamate / metabolism
  • Receptors, N-Methyl-D-Aspartate / drug effects
  • Receptors, N-Methyl-D-Aspartate / metabolism
  • Signal Transduction / physiology

Substances

  • Carrier Proteins
  • Homer Scaffolding Proteins
  • Neuropeptides
  • Receptors, Drug
  • Receptors, Glutamate
  • Receptors, N-Methyl-D-Aspartate
  • GTP-Binding Proteins