Atrasentan Abbott

Curr Opin Investig Drugs. 2002 Aug;3(8):1240-8.

Abstract

Atrasentan is a selective endothelin ET(A) receptor antagonist under development by Abbott for the potential treatment of cancer, particularly prostate cancer, for which it is in phase III trials [413197]. In July 2002, phase II trials for renal, ovarian, lung, colorectal, breast and brain cancers were being initiated [457800]. Atrasentan has been granted Fast Track status, allowing for a rolling NDA [414666], [443479]; the company was planning to begin filing for prostate cancer in late 2003. Atrasentan has also been in phase I trials for hypertension [319405], [326268], but development for this indication had been halted by 2001 [407049].

Publication types

  • Review

MeSH terms

  • Animals
  • Antineoplastic Agents / adverse effects
  • Antineoplastic Agents / chemical synthesis
  • Antineoplastic Agents / metabolism
  • Antineoplastic Agents / pharmacology
  • Antineoplastic Agents / therapeutic use*
  • Atrasentan
  • Cardiovascular System / drug effects
  • Contraindications
  • Endothelin Receptor Antagonists*
  • Humans
  • Male
  • Prostatic Neoplasms / drug therapy*
  • Pyrrolidines*
  • Receptor, Endothelin A
  • Receptors, Endothelin / metabolism
  • Structure-Activity Relationship

Substances

  • Antineoplastic Agents
  • Endothelin Receptor Antagonists
  • Pyrrolidines
  • Receptor, Endothelin A
  • Receptors, Endothelin
  • Atrasentan