[Synthesis of estrone derivatives containing different halogens and/or heterocyclic moieties]

Acta Pharm Hung. 2001 Dec;71(4):441-7.
[Article in Hungarian]

Abstract

New compounds derived from the 3-methyl and 3-benzyl ethers of a D-secoestrone aldehyde were synthesized. In the presence of different Lewis acids D-homosteroids could form. These reactions which can be explained by an intramolecular Prinstype mechanism follow high stereoselectivity and reactivity and lead to compounds containing 16 beta-oriented halogens in the sterane skeleton. The formation and reaction of the imines derived from the aldehyde and aniline as well as substituted anilines provide a highly efficient access to steroid derivatives. The steroid alkaloids are of pharmacological interest.

Publication types

  • English Abstract
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Estrone / analogs & derivatives*
  • Estrone / chemical synthesis*
  • Halogens*
  • Heterocyclic Compounds*
  • Molecular Structure

Substances

  • Halogens
  • Heterocyclic Compounds
  • Estrone