A novel polymorphism, 70Leu/Phe, disrupts a consensus Leu residue within the leucine-rich repeat sequence of platelet glycoprotein Ibalpha

Thromb Haemost. 2002 May;87(5):867-72.

Abstract

Platelet glycoprotein (GP) Ib/IX/V complex mediates high-shear dependent platelet activation through an interaction with the von Willebrand factor (vWF). All four subunits of the complex have a structural motif, the leucine-rich repeat (LRR) sequence, with leucines in conserved positions. Here we report a new polymorphism, Leu/Phe at residue 70 of GPIbalpha, which disrupts the consensus sequence of the LRR in the vWF binding domain. Genotype frequencies among 142 healthy Japanese subjects were 92.3%, 7.7%, and 0.0%, for the 70Leu/Leu, 70Leu/Phe, and 75Phe/Phe genotypes, respectively. Ristocetin-induced or shear-induced platelet aggregation was not significantly different between the 70Leu/Leu and 70Leu/Phe genotypes. In in vitro studies, a recombinant GPIbalpha fragment with 70Phe (L70F) as compared to that with 70Leu (WT) had low reactivity to anti-GPIbalpha monoclonal antibodies, GUR20-5 and Hip1, both of which recognize conformation-specific epitopes within the 45-kDa domain. Ristocetin-induced 125I-vWF binding to L70F, however, did not differ from that to WT.

MeSH terms

  • Amino Acid Substitution*
  • Animals
  • Antibodies, Monoclonal / immunology
  • Antibody Specificity
  • Asian People / genetics
  • Blood Platelets / immunology
  • CHO Cells
  • Consensus Sequence
  • Cricetinae
  • Cricetulus
  • Epitopes / chemistry
  • Epitopes / genetics
  • Epitopes / immunology
  • Gene Frequency
  • Genotype
  • Humans
  • Japan
  • Leucine
  • Mutation, Missense*
  • Peptide Fragments / immunology
  • Platelet Aggregation / drug effects
  • Platelet Glycoprotein GPIb-IX Complex / chemistry
  • Platelet Glycoprotein GPIb-IX Complex / genetics*
  • Platelet Glycoprotein GPIb-IX Complex / immunology
  • Point Mutation
  • Polymorphism, Genetic*
  • Protein Conformation
  • Protein Subunits
  • Recombinant Fusion Proteins / immunology
  • Repetitive Sequences, Amino Acid / genetics*
  • Ristocetin / pharmacology

Substances

  • Antibodies, Monoclonal
  • Epitopes
  • Peptide Fragments
  • Platelet Glycoprotein GPIb-IX Complex
  • Protein Subunits
  • Recombinant Fusion Proteins
  • Ristocetin
  • Leucine