The effects of phytochemical pesticides on the growth of cultured invertebrate and vertebrate cells

Pest Manag Sci. 2002 Mar;58(3):268-76. doi: 10.1002/ps.449.

Abstract

A range of cultured cells of invertebrate and vertebrate origin was grown in the presence of a number of phytochemical pesticides to test the effect of the latter on cell proliferation. The main observation was that azadirachtin was a potent inhibitor of insect cell replication, with an EC50 of 1.5 x 10(10) M against Spodoptera cells and of 6.3 x 10(9) M against Aedes albopictus cells, whilst affecting mammalian cells only at high concentrations (> 10(-4) M). As expected, the other phytochemical pesticides, except for rotenone, had little effect on the growth of the cultured cells. Rotenone was highly effective in inhibiting the growth of insect cells (EC50:10(-8) M) but slightly less toxic towards mammalian cells (EC50:2 x 10(-7) M). Neem terpenoids other than azadirachtin and those very similar in structure significantly inhibited growth of the cell cultures, but to a lesser degree. The major neem seed terpenoids, nimbin and salannin, for example, inhibited insect cell growth by 23% and 15%, respectively.

MeSH terms

  • Animals
  • Cell Division / drug effects
  • Cell Line
  • Cells, Cultured
  • Chrysanthemum cinerariifolium / chemistry
  • Chrysanthemum cinerariifolium / toxicity
  • Diterpenes / chemistry
  • Diterpenes / toxicity
  • Dose-Response Relationship, Drug
  • Humans
  • Insecta / cytology
  • Insecta / drug effects
  • Insecta / growth & development
  • Insecticides / chemistry
  • Insecticides / toxicity*
  • Invertebrates / cytology
  • Invertebrates / drug effects*
  • Invertebrates / growth & development
  • Limonene
  • Limonins*
  • Molecular Structure
  • Rotenone / chemistry
  • Rotenone / toxicity
  • Terpenes / chemistry
  • Terpenes / toxicity
  • Triterpenes / chemistry
  • Triterpenes / toxicity
  • Tumor Cells, Cultured / cytology
  • Tumor Cells, Cultured / drug effects

Substances

  • Diterpenes
  • Insecticides
  • Limonins
  • Terpenes
  • Triterpenes
  • Rotenone
  • salannin
  • Limonene
  • nimbin
  • azadirachtin