Involvement of CDC25Mm/Ras-GRF1-dependent signaling in the control of neuronal excitability

Mol Cell Neurosci. 2001 Dec;18(6):691-701. doi: 10.1006/mcne.2001.1050.

Abstract

Ras-GRF1 is a neuron-specific guanine nucleotide exchange factor for Ras proteins. Mice lacking Ras-GRF1 (-/-) are severely impaired in amygdala-dependent long-term synaptic plasticity and show higher basal synaptic activity at both amygdala and hippocampal synapses (Brambilla et al., 1997). In the present study we investigated the effects of Ras-GRF1 deletion on hippocampal neuronal excitability. Electrophysiological analysis of both primary cultured neurons and adult hippocampal slices indicated that Ras-GRF1-/- mice displayed neuronal hyperexcitability. Ras-GRF1-/- hippocampal neurons showed increased spontaneous activity and depolarized resting membrane potential, together with a higher firing rate in response to injected current. Changes in the intrinsic excitability of Ras-GRF1-/- neurons can entail these phenomena, suggesting that Ras-GRF1 deficiency might alter the balance between ionic conductances. In addition, we showed that mice lacking Ras-GRF1 displayed a higher seizure susceptibility following acute administration of convulsant drugs. Taken together, these results demonstrated a role for Ras-GRF1 in neuronal excitability.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Action Potentials / drug effects
  • Action Potentials / physiology*
  • Animals
  • Electric Stimulation
  • Excitatory Amino Acid Antagonists / pharmacology
  • Excitatory Postsynaptic Potentials / drug effects
  • Excitatory Postsynaptic Potentials / physiology
  • Female
  • Genetic Predisposition to Disease / genetics
  • Glutamate Decarboxylase / metabolism
  • Hippocampus / cytology
  • Hippocampus / drug effects
  • Hippocampus / metabolism*
  • Isoenzymes / metabolism
  • Male
  • Mice
  • Mice, Knockout
  • Nerve Net / cytology
  • Nerve Net / drug effects
  • Nerve Net / metabolism
  • Patch-Clamp Techniques
  • Pyramidal Cells / cytology
  • Pyramidal Cells / drug effects
  • Pyramidal Cells / metabolism*
  • Seizures / chemically induced
  • Seizures / genetics
  • Seizures / metabolism
  • Synaptic Transmission / drug effects
  • Synaptic Transmission / physiology
  • Synaptophysin / metabolism
  • Tetrodotoxin / pharmacology
  • ras-GRF1 / deficiency*
  • ras-GRF1 / genetics

Substances

  • Excitatory Amino Acid Antagonists
  • Isoenzymes
  • Synaptophysin
  • ras-GRF1
  • Tetrodotoxin
  • Glutamate Decarboxylase
  • glutamate decarboxylase 1