Cysteinyl-leukotriene release test (CAST) in the diagnosis of immediate drug reactions

Allergy. 2001 Jul;56(7):688-92. doi: 10.1034/j.1398-9995.2001.00103.x.

Abstract

Background: The diagnosis of allergic reactions to drugs is difficult. Most skin tests are not standardized, and in vitro tests are needed to avoid provocation tests. Cross-linking of IgE on basophils is known to cause the release of both cysteinyl leukotriene (Cys-LT) and histamine. We aimed to evaluate the diagnostic utility (sensitivity, specificity, and efficiency) of measurement of sulfidoleukotrienes in drug allergy.

Methods: We performed a prospective study in 55 patients with proven immediate adverse reactions to drugs (30 to beta-lactams, six to acetaminophen, and 19 to aspirin) and 64 drug-exposed nonallergic controls. Positive diagnosis was established by history, skin tests, and, if needed, oral provocation tests. Cys-LT release was determined after drug-allergen stimulation by the cellular antigen stimulation test (CAST(R)) technique. Histamine release was also assessed on the same samples by enzyme immunoassay. Spontaneous and anti-FcepsilonRIalpha-induced mediator release was also studied in all subjects. Sensitivity, specificity, and efficiency were calculated.

Results: Net Cys-LT release was over the maximal threshold given by the manufacturer in 19/55 patients and in 9/64 controls. Net histamine release was over 5% of total histamine content in 28/55 patients and 34/64 controls. The efficiency of both tests was low.

Conclusion: Thus, in most cases, the in vitro Cys-LT test has little or no diagnostic utility and is not superior to histamine release.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Aged, 80 and over
  • Child
  • Cysteine / metabolism*
  • Diagnostic Techniques and Procedures
  • Drug Hypersensitivity / diagnosis*
  • Female
  • Histamine Release* / physiology
  • Humans
  • Hypersensitivity, Immediate / diagnosis*
  • Inflammation Mediators*
  • Leukotrienes / metabolism*
  • Male
  • Methods
  • Middle Aged
  • Pilot Projects
  • Sensitivity and Specificity
  • Skin Tests / methods

Substances

  • Inflammation Mediators
  • Leukotrienes
  • cysteinyl-leukotriene
  • Cysteine