Regio-reactive resin: a platform for orthogonal loading using the polymer backbone and cross-linker

Bioorg Med Chem Lett. 2001 Jun 18;11(12):1507-9. doi: 10.1016/s0960-894x(01)00152-4.

Abstract

A new support for solid-phase combinatorial organic synthesis has been developed, which we term a regio-reactive resin (R(3)-resin). The resin is based on a unique hydroxyl-functionalized cross-linker readily synthesized in two steps starting from 4-hydroxybenzaldehyde. The cross-linker's ease of synthesis and high purity enables the preparation of gel-type resins with regio-reactive orthogonal loading sites. The resin's swelling properties were investigated, and its potential utility was demonstrated via orthogonal reactivity of the pendant and cross-linker sites.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Absorption
  • Alcohols / chemistry
  • Cross-Linking Reagents / chemistry
  • Polystyrenes / chemistry
  • Resins, Plant / chemical synthesis*
  • Resins, Plant / chemistry
  • Water

Substances

  • Alcohols
  • Cross-Linking Reagents
  • Polystyrenes
  • Resins, Plant
  • Water