Localization of the ribosomal protection protein Tet(O) on the ribosome and the mechanism of tetracycline resistance

Mol Cell. 2001 May;7(5):1037-45. doi: 10.1016/s1097-2765(01)00238-6.

Abstract

Tet(O) belongs to a class of ribosomal protection proteins that mediate tetracycline resistance. It is a G protein that shows significant sequence similarity to elongation factor EF-G. Here we present a cryo-electron microscopic reconstruction, at 16 A resolution, of its complex with the E. coli 70S ribosome. Tet(O) was bound in the presence of a noncleavable GTP analog to programmed ribosomal complexes carrying fMet-tRNA in the P site. Tet(O) is directly visible as a mass close to the A-site region, similar in shape and binding position to EF-G. However, there are important differences. One of them is the different location of the tip of domain IV, which in the Tet(O) case, does not overlap with the ribosomal A site but is directly adjacent to the primary tetracycline binding site. Our findings give insights into the mechanism of tetracycline resistance.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Bacterial Proteins / chemistry
  • Bacterial Proteins / metabolism*
  • Bacterial Proteins / pharmacology
  • Binding Sites
  • Carrier Proteins*
  • Cryoelectron Microscopy
  • Escherichia coli / chemistry
  • Models, Molecular
  • Molecular Conformation
  • Protein Biosynthesis / drug effects
  • Protein Structure, Tertiary
  • RNA-Binding Proteins / chemistry
  • RNA-Binding Proteins / metabolism
  • RNA-Binding Proteins / pharmacology
  • Ribosomes / chemistry*
  • Ribosomes / metabolism
  • Tetracycline Resistance / physiology*

Substances

  • Bacterial Proteins
  • Carrier Proteins
  • RNA-Binding Proteins
  • Tet O resistance protein, Bacteria