Abstract
A novel series of imidazolidinone-based matrix metalloproteinase (MMP) inhibitors was discovered by structural modification of pyrrolidinone la. Potent inhibition of MMP-13 was exhibited by the analogues having 4-(4-fluorophenoxy)phenyl (4a, IC50 = 3 nM) and 4-(naphth-2-yloxy)phenyl (4h, IC50 = 4 nM) as P1' groups.
MeSH terms
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Amides / chemical synthesis*
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Amides / pharmacology*
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Carboxylic Acids / chemical synthesis*
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Carboxylic Acids / pharmacology*
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Drug Design
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Enzyme Inhibitors / chemical synthesis*
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Enzyme Inhibitors / pharmacology
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Imidazoles / chemical synthesis*
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Imidazoles / pharmacology*
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Matrix Metalloproteinase 13
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Matrix Metalloproteinase Inhibitors*
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Stereoisomerism
Substances
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Amides
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Carboxylic Acids
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Enzyme Inhibitors
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Imidazoles
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Matrix Metalloproteinase Inhibitors
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Matrix Metalloproteinase 13