[Spironolactone ameliorates rat pulmonary fibrosis induced by bleomycin A5]

Zhonghua Jie He He Hu Xi Za Zhi. 1998 May;21(5):300-2.
[Article in Chinese]

Abstract

Objective: The purpose of this study was to investigate the role of aldosterone in pulmonary fibrosis and the protective effect of anti-aldosterone treatment.

Method: Rats were divided into control, fibrosis and treatment groups; rat pulmonary fibrosis was induced by endotracheal injection of bleomycin A5 and spironolactone was given 100 mg/kg daily in drinking water to treatment group. 28 days later, plasma, bronchoalveolar lavage fluid(BALF) and tissue aldosterone concentration, as well as lung collagen levels, were determined.

Result: Plasma aldosterone was higher in fibrosis group than that in control group(469 +/- 161 pg/ml and 319 +/- 115 pg/ml, respectively), but without significant difference (P > 0.05); spironolactone could ameliorate the extent of pulmonary fibrosis, the level of lung collagen was 25% less than that of fibrosis group (3.4 +/- 0.5 mg/g lung and 4.6 +/- 1.2 mg/g lung, respectively; q = 3.7893, P < 0.05), and the level of lung protein was 22% less (50 +/- 4 mg/g lung and 65 +/- 6 mg/g lung, respectively; P < 0.01).

Conclusion: Spironolactone had some protective effects on pulmonary fibrosis, and aldosterone might play a role in the development of pulmonary fibrosis.

MeSH terms

  • Aldosterone / metabolism*
  • Animals
  • Bleomycin / analogs & derivatives*
  • Bronchoalveolar Lavage Fluid
  • Collagen / metabolism
  • Lung / metabolism
  • Lung / pathology*
  • Male
  • Mineralocorticoid Receptor Antagonists / pharmacology
  • Pulmonary Fibrosis / chemically induced
  • Pulmonary Fibrosis / metabolism
  • Pulmonary Fibrosis / pathology*
  • Rats
  • Rats, Wistar
  • Spironolactone / pharmacology*

Substances

  • Mineralocorticoid Receptor Antagonists
  • Bleomycin
  • Spironolactone
  • Aldosterone
  • bleomycetin
  • Collagen