Synthesis of new optically active propargylic fluorides and application to the enantioselective synthesis of monofluorinated analogues of fatty acid metabolites

J Org Chem. 2001 May 4;66(9):3146-51. doi: 10.1021/jo010056r.

Abstract

A new approach to obtain optically active unsaturated or polyunsaturated systems with a single fluorine atom in an allylic or propargylic position is reported. Central to this strategy is the high regio- and stereocontrol observed during the fluorination of propargylic alcohols allowing a short and efficient synthesis of 1. Further, simple functional group transformations gave the enals 2 and 3. These three key intermediates were used for the preparation of optically active monofluorinated analogues of fatty acid metabolites.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alkanes / chemistry*
  • Chromatography, Thin Layer
  • Fatty Acids / chemistry*
  • Fatty Acids / metabolism
  • Fatty Acids, Unsaturated / chemistry
  • Fluorides / chemistry*
  • Indicators and Reagents
  • Magnetic Resonance Spectroscopy
  • Spectrophotometry, Ultraviolet
  • Stereoisomerism

Substances

  • Alkanes
  • Fatty Acids
  • Fatty Acids, Unsaturated
  • Indicators and Reagents
  • Fluorides