Prednisolone suppresses ischemia-reperfusion injury of the rat liver by reducing cytokine production and calpain mu activation

J Hepatol. 2001 Feb;34(2):278-83. doi: 10.1016/s0168-8278(00)00017-9.

Abstract

Background: We investigated the effects of prednisolone on cytokine production and calpain mu activation during hepatic ischemia-reperfusion (IR) injury.

Methods: The hilar area of the left lateral and median lobes of rat liver was clamped for 60 min. Prednisolone was administered at 1.0, 3.0, or 10 mg/kg at 30 min before ischemia. In addition to biochemical and microscopic analyses, IL-beta and TNF-alpha production was evaluated by RT-PCR. Calpain mu activation and talin degradation were determined by Western blotting, using specific antibodies.

Results: In the control and prednisolone (1.0 mg/kg) groups, serum AST and ALT levels were elevated, and cell membrane bleb formation was observed after 2 h of reperfusion. Moreover, calpain mu activation, talin degradation, and overexpression of IL-beta and TNF-alpha mRNAs were detected. Infusion of prednisolone at 3.0 or 10 mg/kg significantly suppressed biochemical and microscopic changes. At 10 mg/kg, prednisolone markedly suppressed IL-beta and TNF-alpha transcription and calpain mu activation and talin degradation, consistent with the improved 7-day survival after total hepatic ischemia (75% vs. 25% in control group, P = 0.039).

Conclusions: Cytoprotective effect of prednisolone in hepatic IR injury was closely associated with suppression of IL-beta/TNF-alpha production and calpain mu activation.

MeSH terms

  • Alanine Transaminase / blood
  • Animals
  • Aspartate Aminotransferases / blood
  • Base Sequence
  • Calpain / metabolism*
  • Cytokines / biosynthesis*
  • Cytokines / genetics
  • DNA Primers / genetics
  • Enzyme Activation / drug effects
  • Interleukin-1 / biosynthesis
  • Interleukin-1 / genetics
  • Liver / blood supply*
  • Liver / drug effects
  • Liver / injuries*
  • Liver / pathology
  • Male
  • Prednisolone / administration & dosage
  • Prednisolone / pharmacology*
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • Rats
  • Rats, Wistar
  • Reperfusion Injury / immunology
  • Reperfusion Injury / metabolism
  • Reperfusion Injury / pathology
  • Reperfusion Injury / prevention & control*
  • Talin / metabolism
  • Tumor Necrosis Factor-alpha / biosynthesis
  • Tumor Necrosis Factor-alpha / genetics

Substances

  • Cytokines
  • DNA Primers
  • Interleukin-1
  • RNA, Messenger
  • Talin
  • Tumor Necrosis Factor-alpha
  • Prednisolone
  • Aspartate Aminotransferases
  • Alanine Transaminase
  • Calpain