Ca(2+) sensors of L-type Ca(2+) channel

FEBS Lett. 2000 Dec 29;487(2):301-6. doi: 10.1016/s0014-5793(00)02361-9.

Abstract

Ca(2+)-induced inactivation of L-type Ca(2+) is differentially mediated by two C-terminal motifs of the alpha(1C) subunit, L (1572-1587) and K (1599-1651) implicated for calmodulin binding. We found that motif L is composed of a highly selective Ca(2+) sensor and an adjacent Ca(2+)-independent tethering site for calmodulin. The Ca(2+) sensor contributes to higher Ca(2+) sensitivity of the motif L complex with calmodulin. Since only combined mutation of both sites removes Ca(2+)-dependent current decay, the two-site modulation by Ca(2+) and calmodulin may underlie Ca(2+)-induced inactivation of the channel.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Binding Sites
  • Calcium / metabolism*
  • Calcium Channels, L-Type / chemistry*
  • Calcium Channels, L-Type / genetics
  • Calcium Channels, L-Type / physiology*
  • Calmodulin / metabolism*
  • Cell Line
  • Glutathione Transferase / genetics
  • Kinetics
  • Membrane Potentials / physiology
  • Molecular Sequence Data
  • Recombinant Fusion Proteins / chemistry
  • Recombinant Fusion Proteins / metabolism
  • Transfection

Substances

  • Calcium Channels, L-Type
  • Calmodulin
  • Recombinant Fusion Proteins
  • Glutathione Transferase
  • Calcium