Deacetylase activity associates with topoisomerase II and is necessary for etoposide-induced apoptosis

J Biol Chem. 2001 Feb 16;276(7):4539-42. doi: 10.1074/jbc.C000824200. Epub 2001 Jan 2.

Abstract

DNA topoisomerase II (topo II) is a ubiquitous nuclear enzyme that is involved in DNA replication, transcription, chromosome segregation, and apoptosis. Here we show by immunoprecipitation, pull down with glutathione S-transferase fusion proteins, and yeast two-hybrid analysis that both topo IIalpha and -beta physically interact with the histone deacetylase HDAC1. The in vitro DNA decatenation activity of recombinant topo IIalpha and -beta is inhibited by association with catalytically inactive, recombinant HDAC1. We provide evidence for the in vivo significance of the topo II-HDAC1 association, showing that inhibition of HDAC activity with trichostatin A suppresses apoptosis induced by the topo II poison etoposide, but not by the topoisomerase I inhibitor camptothecin. We suggest that chromatin remodeling by an HDAC-containing complex facilitates both topo II-catalyzed DNA rearrangement and etoposide-induced DNA damage in vivo.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoptosis*
  • DNA Topoisomerases, Type II / metabolism*
  • Enzyme Inhibitors / pharmacology
  • Etoposide / pharmacology*
  • HL-60 Cells
  • HeLa Cells
  • Histone Deacetylase 1
  • Histone Deacetylase Inhibitors
  • Histone Deacetylases / metabolism*
  • Humans
  • Hydroxamic Acids / pharmacology
  • Precipitin Tests
  • Two-Hybrid System Techniques

Substances

  • Enzyme Inhibitors
  • Histone Deacetylase Inhibitors
  • Hydroxamic Acids
  • trichostatin A
  • Etoposide
  • HDAC1 protein, human
  • Histone Deacetylase 1
  • Histone Deacetylases
  • DNA Topoisomerases, Type II