Cardiovascular effects of 3,4-methylenedioxymethamphetamine. A double-blind, placebo-controlled trial

Ann Intern Med. 2000 Dec 19;133(12):969-73. doi: 10.7326/0003-4819-133-12-200012190-00012.

Abstract

Background: The psychoactive stimulant 3, 4-methylenedioxymethamphetamine (MDMA), also known as "ecstasy," is widely used in nonmedical settings. Little is known about its cardiovascular effects.

Objective: To evaluate the acute cardiovascular effects of MDMA by using transthoracic two-dimensional and Doppler echocardiography.

Design: Four-session, ascending-dose, double-blind, placebo-controlled trial.

Setting: Urban hospital.

Patients: Eight healthy adults who self-reported MDMA use.

Intervention: Echocardiographic effects of dobutamine (5, 20, and 40 microg/kg of body weight per minute) were measured in a preliminary session. Oral MDMA (0.5 and 1.5 mg/kg of body weight) or placebo was administered 1 hour before echocardiographic measurements in three weekly sessions.

Measurements: Heart rate and blood pressure were measured at regular intervals before and after MDMA administration. Echocardiographic measures of stroke volume, ejection fraction, cardiac output, and meridional wall stress were obtained 1 hour after MDMA administration and during dobutamine infusions.

Results: At a dose of 1.5 mg/kg, MDMA increased mean heart rate (by 28 beats/min), systolic blood pressure (by 25 mm Hg), diastolic blood pressure (by 7 mm Hg), and cardiac output (by 2 L/min). The effects of MDMA were similar to those of dobutamine, 20 and 40 microg/kg per minute. Inotropism, measured by using meridional wall stress corrected for ejection fraction, decreased after administration of dobutamine, 40 microg/kg per minute, but did not change after either dose of MDMA.

Conclusions: Modest oral doses of MDMA increase heart rate, blood pressure, and myocardial oxygen consumption in a magnitude similar to dobutamine, 20 to 40 microg/kg per minute. In contrast to dobutamine, MDMA has no measurable inotropic effects.

Publication types

  • Clinical Trial
  • Controlled Clinical Trial
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Administration, Oral
  • Adult
  • Analysis of Variance
  • Blood Pressure / drug effects
  • Cardiac Output / drug effects
  • Dose-Response Relationship, Drug
  • Double-Blind Method
  • Echocardiography, Doppler
  • Female
  • Hallucinogens / administration & dosage
  • Hallucinogens / adverse effects*
  • Heart Rate / drug effects
  • Hemodynamics / drug effects*
  • Humans
  • Male
  • N-Methyl-3,4-methylenedioxyamphetamine / administration & dosage
  • N-Methyl-3,4-methylenedioxyamphetamine / adverse effects*
  • Oxygen Consumption / drug effects
  • Stroke Volume / drug effects

Substances

  • Hallucinogens
  • N-Methyl-3,4-methylenedioxyamphetamine