Differential effects of K(+) channel blockers on frequency-dependent action potential broadening in supraoptic neurons

Brain Res Bull. 2000 Sep 15;53(2):203-9. doi: 10.1016/s0361-9230(00)00335-x.

Abstract

Recordings were made from magnocellular neuroendocrine cells dissociated from the supraoptic nucleus of the adult guinea pig to determine the role of voltage gated K(+) channels in controlling the duration of action potentials and in mediating frequency-dependent action potential broadening exhibited by these neurons. The K(+) channel blockers charybdotoxin (ChTx), tetraethylammonium (TEA), and 4-aminopyridine (4-AP) increased the duration of individual action potentials indicating that multiple types of K(+) channel are important in controlling action potential duration. The effect of these K(+) channel blockers was almost completely reversed by simultaneous blockade of voltage gated Ca(2+) channels with Cd(2+). Frequency-dependent action potential broadening was exhibited by these neurons during trains of action potentials elicited by membrane depolarizing current pulses presented at 10 Hz but not at 1 Hz. 4-AP but not ChTx or TEA inhibited frequency-dependent action potential broadening indicating that frequency-dependent action potential broadening is dependent on increasing steady-state inactivation of A-type K(+) channels (which are blocked by 4-AP). A model of differential contributions of voltage gated K(+) channels and voltage gated Ca(2+) channels to frequency-dependent action potential broadening, in which an increase of Ca(2+) current during each successive action potential is permitted as a result of the increasing steady-state inactivation of A-type K(+) channels, is presented.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 4-Aminopyridine / pharmacology
  • Action Potentials / drug effects*
  • Action Potentials / physiology
  • Animals
  • Cadmium Chloride / pharmacology
  • Cells, Cultured
  • Charybdotoxin / pharmacology
  • Guinea Pigs
  • Male
  • Neurons / cytology
  • Neurons / drug effects*
  • Neurons / metabolism
  • Patch-Clamp Techniques
  • Potassium Channel Blockers*
  • Potassium Channels / metabolism
  • Supraoptic Nucleus / cytology
  • Supraoptic Nucleus / drug effects*
  • Supraoptic Nucleus / metabolism
  • Tetraethylammonium / pharmacology

Substances

  • Potassium Channel Blockers
  • Potassium Channels
  • Charybdotoxin
  • Tetraethylammonium
  • 4-Aminopyridine
  • Cadmium Chloride