A fluorescence-quenched chitopentaose for the study of endo-chitinases and chitobiosidases

Eur J Biochem. 2000 Sep;267(17):5593-600. doi: 10.1046/j.1432-1327.2000.01624.x.

Abstract

A new fluorogenic substrate displaying intramolecular fluorescence energy transfer (FRET) has been synthetized from NI,NII,NIII, NIV-tetra-acetyl-chitopentaose. Two molecules, a fluorophore (5-(2-aminoethyl) amino-1-naphtalene-sulfonic acid; EDANS) and a quenching group (dimethylaminophenylazophenyl; DAB) were chemically introduced on to the chitopentaose, one at each end. Among eight enzymes tested, only endo-chitinase and chitobiosidase activities could be specifically assayed by monitoring the variation of fluorescence after enzymatic hydrolysis of this substrate. Chitobiases and N-acetyl-beta-glucosaminidases are not active on the compound, the presence of a bulky chromogenic group at the 2 position of the nonreducing end of the subtrate preventing the binding and thus hydrolysis by these two exo-enzymes. The observation that chitobiosidases are able to hydrolyse a chitooligosaccharide functionalized on both extremities demonstrates the possibility of an endo-action for this class of chitinases, which are generally classified as exo-enzymes. This fluorogenic chitooligosaccharide should prove to be very useful for the detection and the convenient assay of chitinolytic activities at nanomolar concentrations.

MeSH terms

  • Carbohydrate Conformation
  • Carbohydrate Sequence
  • Chitinases / metabolism*
  • Chromatography, High Pressure Liquid
  • Energy Transfer
  • Fluorescence
  • Hexosaminidases / metabolism*
  • Hydrolysis
  • Kinetics
  • Mass Spectrometry
  • Molecular Sequence Data
  • Oligosaccharides / chemistry
  • Oligosaccharides / metabolism*
  • Pyrrolidonecarboxylic Acid / analogs & derivatives
  • Substrate Specificity
  • Thiourea / analogs & derivatives
  • Thiourea / chemistry
  • Thiourea / metabolism*

Substances

  • N(I),N(II),N(III),N(IV)-tetraacetyl-NV-dimethylaminophenylazophenylthioureido-beta-chitopentaosyl-pyroglutamyl amidoethylnaphthalenesulfonic acid
  • Oligosaccharides
  • 1,4-beta-chitobiosidase
  • Hexosaminidases
  • Chitinases
  • Thiourea
  • Pyrrolidonecarboxylic Acid