l-Menthol-induced [Ca2+]i increase and impulses in cultured sensory neurons

Neuroreport. 2000 Jul 14;11(10):2151-5. doi: 10.1097/00001756-200007140-00018.

Abstract

We investigated the effects of l-menthol on cultured dorsal root ganglion (DRG) cells, instead of free nerve endings of sensory fibers. Using Fura-2 microfluorimetry, we identified a few DRG neurons that showed an increase in intracellular free Ca2+ concentration ([Ca2+]i) in response to l-menthol. They made up only 10% of the neurons activated by a high K+ solution. l-Menthol induced the [Ca2+]i increase in a dose-dependent manner, with an EC50 of 37.9 microM and a Hill coefficient of 0.97. A related compound, cyclohexanol, had no effect. When extracellular Ca2+ was removed, l-menthol did not induce the [Ca2+]i increase. Whole-cell current-clamp recordings revealed that l-menthol induced depolarization (13.2 mV, receptor potential) leading to impulses. We conclude that l-menthol induced the impulses through activation of menthol receptors in a small subset of the cultured sensory neurons.

MeSH terms

  • Animals
  • Calcium / metabolism*
  • Cells, Cultured
  • Dose-Response Relationship, Drug
  • Ganglia, Spinal / cytology
  • Ganglia, Spinal / physiology
  • Kinetics
  • Membrane Potentials / drug effects
  • Menthol / pharmacology*
  • Neurons, Afferent / cytology
  • Neurons, Afferent / drug effects
  • Neurons, Afferent / physiology*
  • Patch-Clamp Techniques
  • Potassium / pharmacology
  • Rats
  • Rats, Wistar

Substances

  • Menthol
  • Potassium
  • Calcium