[Role of mutations in the A-subunit of Acholeplasma laidlawii PG-8B topoisomerase IV in formation of resistance to fluoroquinolones]

Mol Gen Mikrobiol Virusol. 2000:(2):30-3.
[Article in Russian]

Abstract

Nucleotide sequence of Acholeplasma laidlawii genome site PG-8B (1000 n.p.), containing topoisomerase IV subunit genes (parE and parC), has been determined. Sequenced genome site contains a gene fragment coding for the C-terminal region of ParE and gene fragment coding for N-terminal region of ParC. Topoisomerase IV subunite genes in A. laidlawii genome are situated near each other and overlapping by 4 nucleotides. Selection in liquid nutrient medium with ascending antibiotic concentrations resulted in derivation of A. laidlawii PG-8B cells resistant to ciprofloxacin, a fluoroquinolone. The resistant clones contain a mutation in the parC QRDR region determining fluoroquinolone resistance: Ser(91) (corresponding to Ser(80) in Escherichia coli ParC) replacement) for Leu.

Publication types

  • English Abstract

MeSH terms

  • Acholeplasma laidlawii / enzymology*
  • Amino Acid Sequence
  • Anti-Infective Agents / pharmacology*
  • Base Sequence
  • DNA Primers
  • DNA Topoisomerase IV
  • DNA Topoisomerases, Type II / chemistry
  • DNA Topoisomerases, Type II / genetics*
  • Drug Resistance, Microbial / genetics
  • Fluoroquinolones
  • Molecular Sequence Data
  • Mutation*
  • Sequence Homology, Amino Acid

Substances

  • Anti-Infective Agents
  • DNA Primers
  • Fluoroquinolones
  • DNA Topoisomerase IV
  • DNA Topoisomerases, Type II