Mechanisms underlying regulated CFTR trafficking

Med Clin North Am. 2000 May;84(3):633-40, ix-x. doi: 10.1016/s0025-7125(05)70246-7.

Abstract

Stimulation of membrane capacitance and cell surface labeling of epitope-tagged CFTR provide evidence of cAMP-regulated CFTR trafficking. Co-expression of syntaxin 1A inhibits cAMP-stimulated current and capacitance changes in CFTR expressing cells and blocks cAMP-induced increases in cell surface CFTR. Inhibition of CFTR trafficking by syntaxin over-expression suggests a role for SNARE proteins in this process. CFTR phosphorylation may alter physical interactions with SNARE proteins to regulate plasma membrane CFTR density.

Publication types

  • Review

MeSH terms

  • Cyclic AMP / physiology
  • Cystic Fibrosis / genetics*
  • Cystic Fibrosis Transmembrane Conductance Regulator / genetics*
  • Gene Expression Regulation / physiology
  • Humans
  • Membrane Proteins / genetics
  • Qa-SNARE Proteins
  • Syntaxin 1

Substances

  • CFTR protein, human
  • Membrane Proteins
  • Qa-SNARE Proteins
  • STX1A protein, human
  • Syntaxin 1
  • Cystic Fibrosis Transmembrane Conductance Regulator
  • Cyclic AMP