JunB suppresses cell proliferation by transcriptional activation of p16(INK4a) expression

EMBO J. 2000 Jun 15;19(12):2969-79. doi: 10.1093/emboj/19.12.2969.

Abstract

A role for the transcription factor JunB in proliferation control was investigated in genetically modified mouse fibroblasts. Increased JunB expression induced high levels of the cyclin-dependent kinase inhibitor p16(INK4a), leading to premature senescence in primary cells and reduced proliferation in 3T3 cells, whereas lack of JunB expression results in decreased p16 levels. Furthermore, JunB-mediated p16 induction in 3T3 cells completely abolished cyclin D-associated kinase activity, resulting in reduced pRb hyperphosphorylation and G(1)-phase extension. Moreover, three AP1-like binding sites were identified in the p16 promoter through which JunB directly activates p16 transcription. Elevated JunB expression in 3T3 cells also inhibited Ras- and Src-mediated transformation and tumour growth in vivo. The suppressive effect of JunB on cell proliferation was shown to be dependent on p16 since it did not occur in INK4a(-/-) fibroblasts that lack both p16 and p19(ARF). These results demonstrate that p16 is a direct transcriptional target gene of JunB and identify JunB as a negative regulator of cell proliferation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Carrier Proteins / biosynthesis*
  • Carrier Proteins / genetics
  • Cell Cycle / physiology*
  • Cell Transformation, Neoplastic
  • Cells, Cultured
  • Cellular Senescence
  • Cyclin D
  • Cyclin-Dependent Kinase Inhibitor p16
  • Cyclin-Dependent Kinases / antagonists & inhibitors*
  • Cyclins
  • Fibroblasts / cytology
  • G1 Phase
  • Mice
  • Mice, Transgenic
  • Oncogene Protein p21(ras)
  • Oncogene Protein pp60(v-src)
  • Promoter Regions, Genetic
  • Protein Kinases
  • Proto-Oncogene Proteins c-jun / genetics
  • Proto-Oncogene Proteins c-jun / metabolism*
  • Transcription Factor AP-1 / metabolism*
  • Transcriptional Activation

Substances

  • Carrier Proteins
  • Cyclin D
  • Cyclin-Dependent Kinase Inhibitor p16
  • Cyclins
  • Proto-Oncogene Proteins c-jun
  • Transcription Factor AP-1
  • Protein Kinases
  • Oncogene Protein pp60(v-src)
  • Cyclin-Dependent Kinases
  • Oncogene Protein p21(ras)