[The antimutagenic activity of afobazol studied in vivo]

Eksp Klin Farmakol. 2000 Mar-Apr;63(2):57-9.
[Article in Russian]

Abstract

The chromosome aberration assay in the bone marrow cells of C57B1/6 mice showed that the new 2-mercaptobenzimidazole derivative afobazole(1-100 mg/kg) prevented manifestations of the clastogenic effects of dioxidine (100 mg/kg, i.p.) over a period of 24 h and reduced by 44-75% the cytogenetic effect of dioxidine (300 mg/kg, i.p.). The same doses of afobazole produced a statistically significant decrease in the cyclophosphamide (20 mg/kg, i.p.) damage over a period of 24 h. Afobazole showed no inherent mutagen activity and did not potentiate the effects of mutagens studied.

MeSH terms

  • Animals
  • Anti-Anxiety Agents / pharmacology*
  • Antimutagenic Agents / pharmacology*
  • Benzimidazoles / pharmacology*
  • Bone Marrow Cells / drug effects
  • Chromosome Aberrations
  • Cyclophosphamide / toxicity
  • Dose-Response Relationship, Drug
  • Drug Interactions
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Morpholines / pharmacology*
  • Mutagens / toxicity
  • Quinoxalines / toxicity

Substances

  • 2-((2-morpholino)ethylthio)-5-ethoxybenzimidazole
  • Anti-Anxiety Agents
  • Antimutagenic Agents
  • Benzimidazoles
  • Morpholines
  • Mutagens
  • Quinoxalines
  • dioxidine
  • Cyclophosphamide