Depletion of cellular protein thiols as an indicator of arylation in isolated trout hepatocytes exposed to 1,4-benzoquinone

Toxicol Sci. 2000 Jun;55(2):327-34. doi: 10.1093/toxsci/55.2.327.

Abstract

A method to measure protein thiols (PrSH), reduced and oxidized, was adapted to determine PrSH depletion in isolated rainbow trout hepatocytes exposed to arylating agent 1,4-benzoquinone (BQ). Toxicant analysis revealed rapid conversion of BQ to 1, 4-hydroquinone (HQ) upon addition to hepatocytes. Hepatocytes exposed to 200 microM BQ+HQ showed 80% decline in glutathione (GSH) (1 h), 30% loss of PrSH (6 h), and no loss of viability (24 h). Recoverable oxidized PrSH was detected only after 24 h (200 microM BQ+HQ). Exposure to 600 microM BQ+HQ caused rapid (10 min) loss of > 90% GSH and > 60% PrSH, with eventual cell death. Half of the PrSH depletion at 6 h observed in hepatocytes exposed to 600 microM BQ+HQ was recoverable by reduction with dithiothreitol. Following the loss of GSH in hepatocytes exposed to 600 microM BQ+HQ, cellular PrSH were susceptible to direct arylation and oxidation. Rainbow trout hepatocytes, which contained 10-fold less GSH than rat cells, had a GSH:PrSH ratio of 1:82 compared with rat ratios of 1:2 to 1:6. The methods reported are useful for further study and discrimination of reactive modes of action needed for prediction of aquatic organism susceptibility to these types of toxicants.

MeSH terms

  • Alkylation
  • Animals
  • Benzoquinones / metabolism
  • Benzoquinones / toxicity*
  • Cell Separation
  • Cell Survival / drug effects
  • Cells, Cultured
  • Dithiothreitol
  • Female
  • Glutathione / metabolism*
  • Glutathione Disulfide / metabolism
  • Hydroquinones / metabolism
  • Liver / cytology
  • Liver / drug effects*
  • Liver / metabolism
  • Male
  • Oncorhynchus mykiss / metabolism*
  • Oxidation-Reduction
  • Sulfhydryl Compounds / metabolism*

Substances

  • Benzoquinones
  • Hydroquinones
  • Sulfhydryl Compounds
  • quinone
  • Glutathione
  • Dithiothreitol
  • Glutathione Disulfide
  • hydroquinone