Asymmetric epoxy cyclohexenyl sulfones: readily accessible progenitors of stereo defined six-carbon arrays

Org Lett. 1999 Aug 12;1(3):355-7. doi: 10.1021/ol990523f.

Abstract

[formula: see text] Enantiopure epoxy vinyl sulfones serve as highly effective substrates for a variety of stereo- and regiospecific oxidation and nucleophilic functionalization reactions. These materials can be easily transformed to cyclic and acyclic six-carbon segments. Nucleophilic epoxidation of 3a,b followed by palladium[0] catalysis enables access to differentially protected arene diols 21 and 22.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Epoxy Compounds / chemistry*
  • Molecular Conformation
  • Stereoisomerism
  • Sulfones / chemistry*

Substances

  • Epoxy Compounds
  • Sulfones