Ketone bodies do not directly alter excitatory or inhibitory hippocampal synaptic transmission

Neurology. 2000 Jan 25;54(2):325-31. doi: 10.1212/wnl.54.2.325.

Abstract

Objective: To determine the effect of the ketone bodies beta-hydroxybutyrate (betaHB) and acetoacetate (AA) on excitatory and inhibitory neurotransmission in the mammalian CNS.

Background: The ketogenic diet is presumed to be an effective anticonvulsant regimen for some children with medically intractable seizures. However, its mechanism of action remains a mystery. According to one hypothesis, ketone bodies have anticonvulsant properties.

Methods: The authors examined the effect of betaHB and AA on excitatory and inhibitory synaptic transmission in rat hippocampal-entorhinal cortex slices and cultured hippocampal neurons. In cultured neurons, their effect was also directly assayed on postsynaptic receptor properties. Finally, their ability to prevent spontaneous seizures was determined in a hippocampal-entorhinal cortex slice model.

Results: betaHB and AA did not alter synaptic transmission in these models.

Conclusions: The anticonvulsant properties of the ketogenic diet do not result from a direct effect of ketone bodies on the primary voltage and ligand gated ion channels mediating excitatory or inhibitory neurotransmission in the hippocampus.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 3-Hydroxybutyric Acid / pharmacology*
  • 4-Aminopyridine
  • Acetoacetates / pharmacology*
  • Animals
  • Cells, Cultured
  • Diet
  • Entorhinal Cortex / cytology
  • Epilepsy / chemically induced
  • Epilepsy / diet therapy
  • Epilepsy / physiopathology
  • Evoked Potentials / drug effects
  • Excitatory Amino Acid Agonists / pharmacology
  • Fasting / physiology
  • Glutamic Acid / pharmacokinetics
  • Glycine / pharmacology
  • Hippocampus / cytology*
  • Kainic Acid / pharmacology
  • Ketosis / etiology
  • Membrane Potentials / drug effects
  • Neural Inhibition / drug effects
  • Neurons / cytology
  • Neurons / drug effects
  • Neurons / physiology*
  • Patch-Clamp Techniques
  • Rats
  • Receptors, AMPA / physiology
  • Receptors, GABA-A / physiology
  • Receptors, Glycine / physiology
  • Receptors, Kainic Acid / physiology
  • Receptors, N-Methyl-D-Aspartate / physiology
  • Stimulation, Chemical
  • Synaptic Membranes / chemistry
  • Synaptic Membranes / drug effects
  • Synaptic Transmission / drug effects*
  • gamma-Aminobutyric Acid / pharmacokinetics

Substances

  • Acetoacetates
  • Excitatory Amino Acid Agonists
  • Receptors, AMPA
  • Receptors, GABA-A
  • Receptors, Glycine
  • Receptors, Kainic Acid
  • Receptors, N-Methyl-D-Aspartate
  • Glutamic Acid
  • gamma-Aminobutyric Acid
  • 4-Aminopyridine
  • Kainic Acid
  • Glycine
  • 3-Hydroxybutyric Acid