Activation of Xenopus eggs by the kinase inhibitor 6-DMAP suggests a differential regulation of cyclin B and p39(mos) proteolysis

Exp Cell Res. 1999 Dec 15;253(2):413-21. doi: 10.1006/excr.1999.4662.

Abstract

In Xenopus eggs, metaphase II arrest is due to the cytostatic factor that maintains a high level of MPF activity. Kinases are important in this phenomenon since p39(mos) and MAPK play a part in the cytostatic activity whereas p34(cdc2) is the catalytic subunit of MPF. Fertilization induces a rise in intracellular calcium leading to egg activation that can be mimicked by calcium-increasing agents such as calcium ionophore. We have performed on Xenopus eggs a biochemical comparison of the effects of the kinase inhibitor 6-DMAP and the calcium ionophore. Both drugs were able to induce pronucleus formation but the underlying molecular events were different. The inactivation of MAPK occurred earlier in eggs exposed to 6-DMAP. Cyclins B1 and B2 were stable and p39(mos) was proteolysed in 6-DMAP-treated eggs while the three proteins underwent degradation in A23187-treated ones. These results suggest a differential regulation of ubiquitin-dependent proteolysis of cyclin B and p39(mos).

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenine / analogs & derivatives*
  • Adenine / pharmacology
  • Animals
  • CDC2 Protein Kinase / analysis
  • CDC2 Protein Kinase / metabolism
  • Calcimycin / pharmacology
  • Calcium / metabolism
  • Cell Nucleus / enzymology
  • Cyclin B / analysis
  • Cyclin B / metabolism*
  • Enzyme Inhibitors / pharmacology*
  • Female
  • Ionophores / pharmacology
  • Metaphase / physiology
  • Mitogen-Activated Protein Kinase 1 / analysis
  • Mitogen-Activated Protein Kinase 1 / metabolism
  • Oocytes / cytology
  • Oocytes / drug effects
  • Oocytes / enzymology*
  • Proto-Oncogene Proteins c-mos / analysis
  • Proto-Oncogene Proteins c-mos / metabolism*
  • Xenopus laevis

Substances

  • Cyclin B
  • Enzyme Inhibitors
  • Ionophores
  • Calcimycin
  • N(6),N(6)-dimethyladenine
  • Proto-Oncogene Proteins c-mos
  • CDC2 Protein Kinase
  • Mitogen-Activated Protein Kinase 1
  • Adenine
  • Calcium