Rat liver in vivo replicative DNA synthesis test for short-term prediction of nongenotoxic (Ames-negative) hepatocarcinogenicity: a collaborative study of the Nongenotoxic Carcinogen Study Group of Japan

Toxicol Lett. 1999 Sep 20;109(1-2):105-14. doi: 10.1016/s0378-4274(99)00129-0.

Abstract

A collaborative study was conducted to evaluate whether a replicative DNA synthesis (RDS) test using the rat liver can detect nongenotoxic (Ames-negative) hepatocarcinogens with three or seven daily administrations at dose-levels effective in long-term bioassays. The assay methods were well-validated by the 14 participants. Of six compounds tested, carbon tetrachloride (50 and 100 mg/kg), clofibrate (125 and 250 mg/kg), diethylstilbestrol (0.125 and 0.25 mg/kg) and urethane (100 mg/kg) gave positive results, methyl carbamate (200 and 400 mg/kg) exerted equivocal effects, and D,L-ethionine (125 mg/kg) failed to elevate RDS. These findings suggest that the RDS test can detect many nongenotoxic rat hepatocarcinogens with short-term administration at dose-levels used in long-term bioassays.

MeSH terms

  • Animals
  • Antimetabolites, Antineoplastic / toxicity
  • Bromodeoxyuridine / toxicity
  • Carcinogenicity Tests / methods*
  • DNA / biosynthesis*
  • DNA Replication / drug effects*
  • Immunohistochemistry
  • Liver / cytology
  • Liver / drug effects
  • Liver / metabolism*
  • Male
  • Mutagenicity Tests / methods*
  • Rats
  • Rats, Inbred F344

Substances

  • Antimetabolites, Antineoplastic
  • DNA
  • Bromodeoxyuridine